Compile Data Set for Download or QSAR
Found 21 of kd data for polymerid = 50006704,50006843
TargetHistone acetyltransferase KAT2A(Homo sapiens (Human))
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50539801(CHEMBL4648912 | US11840533, Compound 70)copy SMILEScopy InChI
Affinity DataKd: <1nMAssay Description:Binding affinity to human partial length GCN5L2 (E726 to K837 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KPPPubMed
TargetHistone acetyltransferase KAT2A(Homo sapiens (Human))
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50573197(CHEMBL4872300)copy SMILES
Affinity DataKd:  44nMAssay Description:Binding affinity to GCN5L2 (unknown origin) by BROMOscan methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5D7GPubMed
TargetHistone acetyltransferase KAT2A(Homo sapiens (Human))
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50512964(CHEMBL4574669)copy SMILEScopy InChI
Affinity DataKd:  105nMAssay Description:Binding affinity to human N-terminal His-tagged GCN5 by isothermal titration calorimetryMore data for this Ligand-Target Pair
TargetHistone acetyltransferase KAT2A(Homo sapiens (Human))
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50514856(CHEMBL4465880)copy SMILEScopy InChI
Affinity DataKd:  158nMAssay Description:Binding affinity to human partial length GCN5L2 (E726 to K837 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN3C7TPubMed
TargetHistone acetyltransferase KAT2A(Homo sapiens (Human))
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM321437((E)-6-(but-2-en-1-yl)-4-(4-(2-hydroxypropan-2-yl)-...)copy SMILEScopy InChI
Affinity DataKd:  160nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetHistone acetyltransferase KAT2A(Homo sapiens (Human))
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50514857(CHEMBL4449894)copy SMILEScopy InChI
Affinity DataKd:  251nMAssay Description:Binding affinity to human partial length GCN5L2 (E726 to K837 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN3C7TPubMed
TargetHistone acetyltransferase KAT2A(Homo sapiens (Human))
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50615275(CHEMBL5282240)copy SMILES
Affinity DataKd:  410nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetHistone acetyltransferase KAT2A(Homo sapiens (Human))
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50514858(CHEMBL4577486)copy SMILEScopy InChI
Affinity DataKd:  501nMAssay Description:Binding affinity to human partial length GCN5L2 (E726 to K837 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN3C7TPubMed
TargetHistone acetyltransferase KAT2A(Homo sapiens (Human))
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM220447(US10633379, Compound X | US9296741, 36)copy SMILEScopy InChI
Affinity DataKd: >1.00E+3nMAssay Description:Inhibition of ADP-induced platelet aggregation in human platelet-rich plasmaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2251MB8PubMed
TargetHistone acetyltransferase KAT2A(Homo sapiens (Human))
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM179481(US9675697, Cpd. No. 73)copy SMILEScopy InChI
Affinity DataKd: >4.00E+3nMAssay Description:Binding affinity to human partial length GCN5L2 (E726 to K837 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3GWNPubMed
TargetHistone acetyltransferase GCN5(Saccharomyces cerevisiae S288c)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50371146(CHEMBL4168633)copy SMILEScopy InChI
Affinity DataKd:  4.20E+3nMAssay Description:Binding affinity to yeast GCN5 (99 to 262 residues) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HPJPubMed
TargetHistone acetyltransferase KAT2A(Homo sapiens (Human))
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50366670(CHEMBL4173488)copy SMILEScopy InChI
Affinity DataKd: >5.00E+3nMAssay Description:Binding affinity to human GCN5L2 (E726 to K837 residues) expressed in bacterial expression system by BROMOScan assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M39B1PubMed
TargetHistone acetyltransferase KAT2A(Homo sapiens (Human))
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM321424(6-[(E)-but-2-enyl]-4-[2,5-dimethoxy-4-(morpholine-...)copy SMILEScopy InChI
Affinity DataKd: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone acetyltransferase KAT2A(Homo sapiens (Human))
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50453949(CHEMBL4208820 | US11247989, Example 87)copy SMILEScopy InChI
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human partial length GCN5L2 (E726 to K837 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6VVZPubMed
TargetHistone acetyltransferase KAT2A(Homo sapiens (Human))
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM249277(US10017501, Compound 1020-18 | US9458145, 1020-18)copy SMILEScopy InChI
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human partial length GCN5L2 (E726 to K837 residues) expressed in bacterial expression system after 1 hr by bromoscan assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7ZZ6PubMed
TargetHistone acetyltransferase KAT2A(Homo sapiens (Human))
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50615276(CHEMBL5270178)copy SMILES
Affinity DataKd: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetHistone acetyltransferase GCN5(Saccharomyces cerevisiae S288c)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50372744(CHEMBL4165080)copy SMILEScopy InChI
Affinity DataKd:  2.62E+4nMAssay Description:Binding affinity to yeast GCN5 (99 to 262 residues) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HPJPubMed
TargetHistone acetyltransferase KAT2A(Homo sapiens (Human))
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50455480(CHEMBL4218735)copy SMILEScopy InChI
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged GCN5L2 expressed in bacteria by BROMOscan methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetHistone acetyltransferase KAT2A(Homo sapiens (Human))
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50098311(CHEMBL3590408)copy SMILES
Affinity DataKd: <1.00E+5nMAssay Description:Binding affinity to KAT2A in human HUT78 cells incubated for 45 mins by mass spectrometry based bromosphere chemoproteomic assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN17Z1PubMed
TargetHistone acetyltransferase KAT2A(Homo sapiens (Human))
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50098305(CHEMBL3590405)copy SMILES
Affinity DataKd: <1.00E+5nMAssay Description:Binding affinity to KAT2A in human HUT78 cells incubated for 45 mins by mass spectrometry based bromosphere chemoproteomic assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN17Z1PubMed
TargetHistone acetyltransferase KAT2A(Homo sapiens (Human))
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50098250(CHEMBL3590389)copy SMILEScopy InChI
Affinity DataKd: <1.00E+5nMAssay Description:Binding affinity to KAT2A in human HUT78 cells incubated for 45 mins by mass spectrometry based bromosphere chemoproteomic assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN17Z1PubMed